PI3Kδ and PI3Kγ as targets for autoimmune and inflammatory diseases

J Med Chem. 2012 Oct 25;55(20):8559-81. doi: 10.1021/jm300847w. Epub 2012 Sep 13.
No abstract available

Publication types

  • Review

MeSH terms

  • Animals
  • Autoimmune Diseases / drug therapy
  • Autoimmune Diseases / enzymology*
  • B-Lymphocytes / enzymology
  • Class Ia Phosphatidylinositol 3-Kinase / chemistry
  • Class Ia Phosphatidylinositol 3-Kinase / metabolism*
  • Class Ib Phosphatidylinositol 3-Kinase / chemistry
  • Class Ib Phosphatidylinositol 3-Kinase / metabolism*
  • Humans
  • Inflammation / drug therapy
  • Inflammation / enzymology*
  • Isoenzymes / antagonists & inhibitors
  • Isoenzymes / metabolism
  • Molecular Targeted Therapy
  • Neutrophils / enzymology
  • Phosphoinositide-3 Kinase Inhibitors*
  • Protein Conformation
  • T-Lymphocytes / enzymology

Substances

  • Isoenzymes
  • Phosphoinositide-3 Kinase Inhibitors
  • Class Ia Phosphatidylinositol 3-Kinase
  • Class Ib Phosphatidylinositol 3-Kinase